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@ARTICLE{Vragniau:120552,
author = {C. Vragniau and J.-M. Hübner$^*$ and P. Beidler and S. Gil
and K. Saydaminova and Z.-Z. Lu and R. Yumul and H. Wang and
M. Richter and P. Sova and C. Drescher and P. Fender and A.
Lieber},
title = {{S}tudies on the {I}nteraction of {T}umor-{D}erived {HD}5
{A}lpha {D}efensins with {A}denoviruses and {I}mplications
for {O}ncolytic {A}denovirus {T}herapy.},
journal = {Journal of virology},
volume = {91},
number = {6},
issn = {1098-5514},
address = {Baltimore, Md.},
publisher = {Soc.},
reportid = {DKFZ-2017-00981},
pages = {e02030-16 -},
year = {2017},
abstract = {Defensins are small antimicrobial peptides capable of
neutralizing human adenovirus (HAdV) in vitro by binding
capsid proteins and blocking endosomal escape of virus. In
humans, the alpha defensin HD5 is produced by specialized
epithelial cells of the gastrointestinal and genito-urinary
tracts. Here, we demonstrate, using patient biopsy
specimens, that HD5 is also expressed as an active, secreted
peptide by epithelial ovarian and lung cancer cells in situ
This finding prompted us to study the role of HD5 in
infection and spread of replication-competent, oncolytic
HAdV type 3 (HAdV3). HAdV3 produces large amounts of
penton-dodecahedra (PtDd), virus-like particles, during
replication. We have previously shown that PtDd are involved
in opening epithelial junctions, thus facilitating lateral
spread of de novo-produced virions. Here, we describe a
second function of PtDd, namely, the blocking of HD5. A
central tool to prove that viral PtDd neutralize HD5 and
support spread of progeny virus was an HAdV3 mutant virus in
which formation of PtDd was disabled (mut-Ad3GFP, where GFP
is green fluorescent protein). We demonstrated that viral
spread of mut-Ad3GFP was blocked by synthetic HD5 whereas
that of the wild-type (wt) form (wt-Ad3GFP) was only
minimally impacted. In human colon cancer Caco-2 cells,
induction of cellular HD5 expression by fibroblast growth
factor 9 (FGF9) significantly inhibited viral spread and
progeny virus production of mut-Ad3GFP but not of wt-Ad3GFP.
Finally, the ectopic expression of HD5 in tumor cells
diminished the in vivo oncolytic activity of mut-Ad3GFP but
not of wt-Ad3GFP. These data suggest a new mechanism of
HAdV3 to overcome innate antiviral host responses. Our study
has implications for oncolytic adenovirus therapy.IMPORTANCE
Previously, it has been reported that human defensin HD5
inactivates specific human adenoviruses by binding to capsid
proteins and blocking endosomal escape of virus. The central
new findings described in our manuscript are the following:
(i) the discovery of a new mechanism used by human
adenovirus serotype 3 to overcome innate antiviral host
responses that is based on the capacity of HAdV3 to produce
subviral penton-dodecahedral particles that act as decoys
for HD5, thus preventing the inactivation of virus progeny
produced upon replication; (ii) the demonstration that
ectopic HD5 expression in cancer cells decreases the
oncolytic efficacy of a serotype 5-based adenovirus vector;
and (iii) the demonstration that epithelial ovarian and lung
cancers express HD5. The study improves our understanding of
how adenoviruses establish infection in epithelial tissues
and has implications for cancer therapy with oncolytic
adenoviruses.},
keywords = {alpha-Defensins (NLM Chemicals) / alpha-defensin 5, human
(NLM Chemicals)},
cin = {B062},
ddc = {570},
cid = {I:(DE-He78)B062-20160331},
pnm = {312 - Functional and structural genomics (POF3-312)},
pid = {G:(DE-HGF)POF3-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:28077642},
pmc = {pmc:PMC5331826},
doi = {10.1128/JVI.02030-16},
url = {https://inrepo02.dkfz.de/record/120552},
}