%0 Journal Article %A von Hagens, Cornelia %A Walter-Sack, Ingeborg %A Goeckenjan, Maren %A Osburg, Julia %A Storch-Hagenlocher, Brigitte %A Sertel, Serkan %A Elsässer, Michael %A Remppis, Bjoern Andrew %A Edler, Lutz %A Munzinger, Judith %A Efferth, Thomas %A Schneeweiss, Andreas %A Strowitzki, Thomas %T Prospective open uncontrolled phase I study to define a well-tolerated dose of oral artesunate as add-on therapy in patients with metastatic breast cancer (ARTIC M33/2). %J Breast cancer research and treatment %V 164 %N 2 %@ 1573-7217 %C Dordrecht [u.a.] %I Springer Science + Business Media B.V. %M DKFZ-2017-01318 %P 359 - 369 %D 2017 %X The antimalarial drug artesunate (ART) is a promising candidate for cancer treatment as it displays anticancer effects in various models. While in short-term treatment of malaria, an excellent safety profile has been found for ART, the potential long-term treatment of cancer patients demands a phase I dose-finding clinical trial determining the daily ART dose which would be well tolerated as add-on therapy.Patients with metastatic breast cancer were to receive either 100 or 150 or 200 mg oral ART daily as add-on to their guideline-based oncological therapy for a study period of four weeks with frequent clinical and laboratory monitoring until 4-8 weeks thereafter. According to the statistical design, recruitment was scheduled in groups of three patients in order not to miss a more than 33 %F PUB:(DE-HGF)16 %9 Journal Article %$ pmid:28439738 %R 10.1007/s10549-017-4261-1 %U https://inrepo02.dkfz.de/record/124441