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@ARTICLE{Hellwig:143312,
author = {M. Hellwig and M. C. Lauffer and M. Bockmayr and M. Spohn
and D. J. Merk and L. Harrison and J. Ahlfeld and A.
Kitowski and J. E. Neumann and J. Ohli and D. Holdhof and J.
Niesen and M. Schoof and M. Kool$^*$ and C. Kraus and C.
Zweier and D. Holmberg and U. Schüller},
title = {{TCF}4 ({E}2-2) harbors tumor suppressive functions in
{SHH} medulloblastoma.},
journal = {Acta neuropathologica},
volume = {137},
number = {4},
issn = {1432-0533},
address = {Heidelberg},
publisher = {Springer},
reportid = {DKFZ-2019-00902},
pages = {657 - 673},
year = {2019},
abstract = {The TCF4 gene encodes for the basic helix-loop-helix
transcription factor 4 (TCF4), which plays an important role
in the development of the central nervous system (CNS).
Haploinsufficiency of TCF4 was found to cause Pitt-Hopkins
syndrome (PTHS), a severe neurodevelopmental disorder.
Recently, the screening of a large cohort of medulloblastoma
(MB), a highly aggressive embryonal brain tumor, revealed
almost $20\%$ of adult patients with MB of the Sonic
hedgehog (SHH) subtype carrying somatic TCF4 mutations.
Interestingly, many of these mutations have previously been
detected as germline mutations in patients with PTHS. We
show here that overexpression of wild-type TCF4 in vitro
significantly suppresses cell proliferation in MB cells,
whereas mutant TCF4 proteins do not to the same extent.
Furthermore, RNA sequencing revealed significant
upregulation of multiple well-known tumor suppressors upon
expression of wild-type TCF4. In vivo, a prenatal knockout
of Tcf4 in mice caused a significant increase in apoptosis
accompanied by a decreased proliferation and failed
migration of cerebellar granule neuron precursor cells
(CGNP), which are thought to be the cells of origin for SHH
MB. In contrast, postnatal in vitro and in vivo knockouts of
Tcf4 with and without an additional constitutive activation
of the SHH pathway led to significantly increased
proliferation of CGNP or MB cells. Finally, publicly
available data from human MB show that relatively low
expression levels of TCF4 significantly correlate with a
worse clinical outcome. These results not only point to
time-specific roles of Tcf4 during cerebellar development
but also suggest a functional linkage between TCF4 mutations
and the formation of SHH MB, proposing that TCF4 acts as a
tumor suppressor during postnatal stages of cerebellar
development.},
cin = {B062 / L101},
ddc = {610},
cid = {I:(DE-He78)B062-20160331 / I:(DE-He78)L101-20160331},
pnm = {312 - Functional and structural genomics (POF3-312)},
pid = {G:(DE-HGF)POF3-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:30830316},
doi = {10.1007/s00401-019-01982-5},
url = {https://inrepo02.dkfz.de/record/143312},
}