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@ARTICLE{AbdulPari:154531,
author = {A. A. Abdul Pari$^*$ and M. Singhal$^*$ and C. Hübers$^*$
and C. Mogler and B. Schieb$^*$ and A. Gampp$^*$ and N.
Gengenbacher$^*$ and L. E. Reynolds and D. Terhardt$^*$ and
C. Géraud and J. Utikal$^*$ and M. Thomas and S. Goerdt and
K. M. Hodivala-Dilke and H. Augustin$^*$ and M. Felcht},
title = {{T}umor cell-derived {A}ngiopoietin-2 promotes metastasis
in melanoma.},
journal = {Cancer research},
volume = {80},
number = {12},
issn = {1538-7445},
address = {Philadelphia, Pa.},
publisher = {AACR},
reportid = {DKFZ-2020-00852},
pages = {2586-2598},
year = {2020},
note = {DKFZ-ZMBH Alliance2020 Jun
15;80(12):2586-2598#EA:A190#LA:A190#},
abstract = {The Angiopoietin (Angpt)-TIE signaling pathway controls
vascular maturation and maintains the quiescent phenotype of
resting vasculature. The contextual agonistic and
antagonistic Tie2 ligand ANGPT2 is believed to be
exclusively produced by endothelial cells, disrupting
constitutive ANGPT1-TIE2 signaling to destabilize the
microvasculature during pathological disorders like
inflammation and cancer. However, scattered reports have
also portrayed tumor cells as a source of ANGPT2. Employing
in situ hybridization-based detection of ANGPT2, we found
strong tumor cell expression of ANGPT2 in a subset of
melanoma patients. Comparative analysis of biopsies revealed
a higher fraction of ANGPT2-expressing tumor cells in
metastatic versus primary sites. Tumor cell-expressed Angpt2
was dispensable for primary tumor growth, yet in-depth
analysis of primary tumors revealed enhanced intratumoral
necrosis upon silencing of tumor cell Angpt2 expression in
the absence of significant immune and vascular alterations.
Global transcriptional profiling of Angpt2-deficient tumor
cells identified perturbations in redox homeostasis and an
increased response to cellular oxidative stress.
Ultrastructural analyses illustrated a significant increase
of dysfunctional mitochondria in Angpt2-silenced tumor
cells, thereby resulting in enhanced ROS production and
downstream MAPK stress signaling. Functionally, enhanced ROS
in Angpt2-silenced tumor cells reduced colonization
potential in vitro and in vivo. Taken together, these
findings uncover the hitherto unappreciated role of tumor
cell-expressed ANGPT2 as an autocrine positive regulator of
metastatic colonization and validate ANGPT2 as a therapeutic
target for a well-defined subset of melanoma patients.},
cin = {A190 / A370 / HD01},
ddc = {610},
cid = {I:(DE-He78)A190-20160331 / I:(DE-He78)A370-20160331 /
I:(DE-He78)HD01-20160331},
pnm = {311 - Signalling pathways, cell and tumor biology
(POF3-311)},
pid = {G:(DE-HGF)POF3-311},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:32303578},
doi = {10.1158/0008-5472.CAN-19-2660},
url = {https://inrepo02.dkfz.de/record/154531},
}