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@ARTICLE{Miele:163162,
author = {E. Miele and A. Po and A. Mastronuzzi and A. Carai and Z.
M. Besharat and N. Pediconi and L. Abballe and G. Catanzaro
and C. Sabato and E. De Smaele and G. Canettieri and L. Di
Marcotullio and A. Vacca and A. Mai and M. Levrero and S. M.
Pfister$^*$ and M. Kool$^*$ and F. Giangaspero and F.
Locatelli and E. Ferretti},
title = {{D}ownregulation of mi{R}-326 and its host gene
β-arrestin1 induces pro survival activity of {E}2{F}1 and
promotes medulloblastoma growth.},
journal = {Molecular oncology},
volume = {15},
number = {2},
issn = {1574-7891},
address = {Hoboken, NJ},
publisher = {John Wiley $\&$ Sons, Inc.},
reportid = {DKFZ-2020-01865},
pages = {523-542},
year = {2021},
note = {2021 Feb;15(2):523-542},
abstract = {Persistent mortality rates of medulloblastoma (MB) and
severe side effects of the current therapies require the
definition of the molecular mechanisms that contribute to
tumor progression. Using cultured MB cancer stem cells and
xenograft tumors generated in mice, we show that low
expression of miR-326 and its host gene β-arrestin1 (ARRB1)
promotes tumor growth enhancing the E2F1 pro-survival
function. Our models revealed that miR-326 and ARRB1 are
controlled by a bivalent domain, since the H3K27me3
repressive mark is found at their regulatory region together
with the activation-associated H3K4me3 mark. High levels of
EZH2, a feature of MB, are responsible for the presence of
H3K27me3. Ectopic expression of miR-326 and ARRB1 provides
hints into how their low levels regulate E2F1 activity.
MiR-326 targets E2F1 mRNA, thereby reducing its protein
levels; ARRB1, triggering E2F1 acetylation, reverses its
function into pro-apoptotic activity. Similar to miR-326 and
ARRB1 overexpression, we also show that EZH2 inhibition
restores miR-326/ARRB1 expression, limiting E2F1
pro-proliferative activity. Our results reveal a new
regulatory molecular axis critical for MB progression.},
cin = {B062},
ddc = {610},
cid = {I:(DE-He78)B062-20160331},
pnm = {312 - Funktionelle und strukturelle Genomforschung
(POF4-312)},
pid = {G:(DE-HGF)POF4-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:32920979},
doi = {10.1002/1878-0261.12800.},
url = {https://inrepo02.dkfz.de/record/163162},
}