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@ARTICLE{Zwicker:166693,
author = {F. Zwicker$^*$ and H. Hauswald and K.-J. Weber and J.
Debus$^*$ and P. Huber$^*$},
title = {{I}n {V}ivo {E}valuation of {C}ombined {CK}2 {I}nhibition
and {I}rradiation in {H}uman {W}i{D}r {T}umours.},
journal = {In vivo},
volume = {35},
number = {1},
issn = {1791-7549},
address = {Kapandriti, Attiki},
publisher = {IIAR},
reportid = {DKFZ-2021-00046},
pages = {111 - 117},
year = {2021},
note = {#EA:E050#LA:E055#},
abstract = {Casein kinase 2 (CK2) which sustains multiple pro-survival
functions in cellular DNA-damage response, is strictly
regulated in normal cells but elevated in cancer. CK2 is
considered as a potential therapeutic target, and its
inhibition has been associated with radiosensitization in
mammalian cells in vitro. Here, we investigated potential
radiosensitization by CK2 inhibition in vivo.The effect of
CK2 inhibition in vivo was investigated in human
WiDr-xenograft tumours grown subcutaneously on BALB/c nu/nu
mice with and without fractionated irradiation. CK2
inhibition was performed using the specific inhibitor
tetra-bromobenzotriazole (TBB). Histological examinations
included staining for apoptosis and double-strand
breaks.Both TBB treatment alone and radiation alone
significantly reduced tumour growth, which was reflected by
increased apoptosis rates. However, TBB treatment did not
boost radiation-induced tumour growth suppression in
combined treatment, although the apoptosis rate increased
and repair of double-strand breaks was reduced. This was in
stark contrast to previous data on in vitro
radiosensitization.The absence of radiosensitization by CK2
inhibition should be investigated in different tumour
models.},
keywords = {CK2 inhibition (Other) / TBB (Other) / human WiDr tumours
(Other) / irradiation (Other) / tetra-bromobenzotriazole
(Other)},
cin = {E050 / E055},
ddc = {610},
cid = {I:(DE-He78)E050-20160331 / I:(DE-He78)E055-20160331},
pnm = {315 - Bildgebung und Radioonkologie (POF4-315)},
pid = {G:(DE-HGF)POF4-315},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:33402456},
doi = {10.21873/invivo.12238},
url = {https://inrepo02.dkfz.de/record/166693},
}