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@ARTICLE{Fresnais:167771,
author = {M. Fresnais and E. Yildirim and S. Karabulut and D. Jäger
and I. Zörnig and J. Benzel$^*$ and K. W. Pajtler$^*$ and
S. M. Pfister$^*$ and J. Burhenne and W. E. Haefeli and R.
Longuespée},
title = {{R}apid {MALDI}-{MS} {A}ssays for {D}rug {Q}uantification
in {B}iological {M}atrices: {L}essons {L}earned, {N}ew
{D}evelopments, and {F}uture {P}erspectives.},
journal = {Molecules},
volume = {26},
number = {5},
issn = {1420-3049},
address = {Basel},
publisher = {MDPI44576},
reportid = {DKFZ-2021-00535},
pages = {1281},
year = {2021},
note = {2021 Feb 26;26(5):1281},
abstract = {Matrix-assisted laser desorption/ionization mass
spectrometry (MALDI-MS) has rarely been used in the field of
therapeutic drug monitoring, partly because of the
complexity of the ionization processes between the compounds
to be quantified and the many MALDI matrices available. The
development of a viable MALDI-MS method that meets
regulatory guidelines for bioanalytical method validation
requires prior knowledge of the suitability of (i) the MALDI
matrix with the analyte class and properties for ionization,
(ii) the crystallization properties of the MALDI matrix with
automation features, and (iii) the MS instrumentation used
to achieve sensitive and specific measurements in order to
determine low pharmacological drug concentrations in
biological matrices. In the present hybrid article/white
paper, we review the developments required for the
establishment of MALDI-MS assays for the quantification of
drugs in tissues and plasma, illustrated with concrete
results for the different steps. We summarize the necessary
parameters that need to be controlled for the successful
development of fully validated MALDI-MS methods according to
regulatory authorities, as well as currently unsolved
problems and promising ways to address them. Finally, we
propose an expert opinion on future perspectives and needs
in order to establish MALDI-MS as a universal method for
therapeutic drug monitoring.},
keywords = {MALDI (Other) / mass spectrometry (Other) / targeted
quantification (Other) / therapeutic drug monitoring
(Other)},
cin = {B062 / HD01},
ddc = {540},
cid = {I:(DE-He78)B062-20160331 / I:(DE-He78)HD01-20160331},
pnm = {312 - Funktionelle und strukturelle Genomforschung
(POF4-312)},
pid = {G:(DE-HGF)POF4-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:33652935},
doi = {10.3390/molecules26051281},
url = {https://inrepo02.dkfz.de/record/167771},
}