% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Feuerecker:275422,
author = {B. Feuerecker$^*$ and C. Kratochwil and H. Ahmadzadehfar
and A. Morgenstern and M. Eiber and K. Herrmann$^*$ and K.
L. Pomykala},
title = {{C}linical {T}ranslation of {T}argeted α-{T}herapy: {A}n
{E}volution or a {R}evolution?},
journal = {Journal of nuclear medicine},
volume = {64},
number = {5},
issn = {0097-9058},
address = {New York, NY},
publisher = {Soc.},
reportid = {DKFZ-2023-00745},
pages = {685-692},
year = {2023},
note = {2023 May;64(5):685-692},
abstract = {The field of radioligand therapy has advanced greatly in
recent years, driven largely by β-emitting therapies
targeting somatostatin receptor-expressing tumors and the
prostate-specific membrane antigen. Now, more clinical
trials are under way to evaluate α-emitting targeted
therapies as potential next-generation theranostics with
even higher efficacy due to their high linear energy and
short range in human tissues. In this review, we summarize
the important studies ranging from the first Food and Drug
Administration-approved α-therapy, 223Ra-dichloride, for
treatment of bone metastases in castration-resistant
prostate cancer, including concepts in clinical translation
such as targeted α-peptide receptor radiotherapy and
225Ac-PSMA-617 for treatment of prostate cancer, innovative
therapeutic models evaluating new targets, and combination
therapies. Targeted α-therapy is one of the most promising
fields in novel targeted cancer therapy, with several early-
and late-stage clinical trials for neuroendocrine tumors and
metastatic prostate cancer already in progress, along with
significant interest and investment in additional
early-phase studies. Together, these studies will help us
understand the short- and long-term toxicity of targeted
α-therapy and potentially identify suitable therapeutic
combination partners.},
subtyp = {Review Article},
keywords = {225Ac (Other) / PSMA-617 (Other) / targeted α-therapy
(Other) / α-emitter (Other)},
cin = {MU01 / ED01},
ddc = {610},
cid = {I:(DE-He78)MU01-20160331 / I:(DE-He78)ED01-20160331},
pnm = {899 - ohne Topic (POF4-899)},
pid = {G:(DE-HGF)POF4-899},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:37055224},
doi = {10.2967/jnumed.122.265353},
url = {https://inrepo02.dkfz.de/record/275422},
}