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@ARTICLE{Dong:275927,
author = {H. Dong and L. Zeng and W. Chen and Q. Zhang and F. Wang
and Y. Wu and B. Cui and J. Qi and X. Zhang and C. Liu and
J. Deng and Y. Yu and C. A. Schmitt$^*$ and J. Du},
title = {{N}6-methyladenine-mediated aberrant activation of the
lnc{RNA} {SOX}2{OT}-{GLI}1 loop promotes non-small-cell lung
cancer stemness.},
journal = {Cell death discovery},
volume = {9},
number = {1},
issn = {2058-7716},
address = {London},
publisher = {Nature Publishing Group},
reportid = {DKFZ-2023-00915},
pages = {149},
year = {2023},
abstract = {Despite the advent of precision medicine and immunotherapy,
mortality due to lung cancer remains high. The sonic
hedgehog (SHH) cascade and its key terminal factor,
glioma-associated oncogene homolog 1 (GLI1), play a pivotal
role in the stemness and drug resistance of lung cancer.
Here, we investigated the molecular mechanism of
non-canonical aberrant GLI1 upregulation. The SHH cascade
was upregulated in stem spheres and chemo-resistant lung
cancer cells and was accountable for drug resistance against
multiple chemotherapy regimens. GLI1 and the long non-coding
RNA SOX2OT were positively regulated, and the GLI1-SOX2OT
loop mediated the proliferation of parental and stem-like
lung cancer cells. Further mechanistic investigation
revealed that SOX2OT facilitated METTL3/14/IGF2BP2-mediated
m6A modification and stabilization of the GLI1 mRNA.
Additionally, SOX2OT upregulated METTL3/14/IGF2BP2 by
sponging miR-186-5p. Functional analysis corroborated that
GLI1 acted as a downstream target of METTL3/14/IGF2BP2, and
GLI1 silencing could block the oncogenicity of lung cancer
stem-like cells. Pharmacological inhibition of the loop
remarkably inhibited the oncogenesis of lung cancer cells in
vivo. Compared with paired adjacent normal tissues, lung
cancer specimens exhibited consistently upregulated
GLI1/SOX2OT/METTL3/14/IGF2BP2. The m6A-modified GLI1-SOX2OT
loop may serve as a potential therapeutic target and
prognostic predictor for lung cancer therapy and diagnosis
in the clinic.},
cin = {BE01},
ddc = {610},
cid = {I:(DE-He78)BE01-20160331},
pnm = {899 - ohne Topic (POF4-899)},
pid = {G:(DE-HGF)POF4-899},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:37149646},
pmc = {pmc:PMC10164154},
doi = {10.1038/s41420-023-01442-w},
url = {https://inrepo02.dkfz.de/record/275927},
}