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@ARTICLE{Beumers:285945,
author = {L. Beumers$^*$ and E.-I. Vlachavas$^*$ and S. Borgoni$^*$
and L. Schwarzmüller$^*$ and L. Penso-Dolfin$^*$ and B.
Michels$^*$ and E. Sofyali$^*$ and S. Burmester$^*$ and D.
Heiss$^*$ and H. Wilhelm$^*$ and Y. Yarden and D. Helm$^*$
and R. Will$^*$ and A. Goncalves$^*$ and S. Wiemann$^*$},
title = {{C}lonal heterogeneity in {ER}+ breast cancer reveals the
proteasome and {PKC} as potential therapeutic targets.},
journal = {npj Breast cancer},
volume = {9},
number = {1},
issn = {2374-4677},
address = {London},
publisher = {Nature Publ. Group},
reportid = {DKFZ-2023-02535},
pages = {97},
year = {2023},
note = {#EA:B050#LA:B050#},
abstract = {Intratumoral heterogeneity impacts the success or failure
of anti-cancer therapies. Here, we investigated the
evolution and mechanistic heterogeneity in clonal
populations of cell models for estrogen receptor positive
breast cancer. To this end, we established barcoded models
of luminal breast cancer and rendered them resistant to
commonly applied first line endocrine therapies. By
isolating single clones from the resistant cell pools and
characterizing replicates of individual clones we observed
inter- (between cell lines) and intra-tumor (between
different clones from the same cell line) heterogeneity.
Molecular characterization at RNA and phospho-proteomic
levels revealed private clonal activation of the unfolded
protein response and respective sensitivity to inhibition of
the proteasome, and potentially shared sensitivities for
repression of protein kinase C. Our in vitro findings are
consistent with tumor-heterogeneity that is observed in
breast cancer patients thus highlighting the need to uncover
heterogeneity at an individual patient level and to adjust
therapies accordingly.},
cin = {B050 / B210 / W120 / W111},
ddc = {610},
cid = {I:(DE-He78)B050-20160331 / I:(DE-He78)B210-20160331 /
I:(DE-He78)W120-20160331 / I:(DE-He78)W111-20160331},
pnm = {312 - Funktionelle und strukturelle Genomforschung
(POF4-312)},
pid = {G:(DE-HGF)POF4-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:38042915},
pmc = {pmc:PMC10693625},
doi = {10.1038/s41523-023-00604-4},
url = {https://inrepo02.dkfz.de/record/285945},
}