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@ARTICLE{Almouhanna:287409,
author = {F. Almouhanna and J. Hess$^*$},
title = {{A}n {ESR}1-{R}elated {G}ene {S}ignature {I}dentifies
{H}ead and {N}eck {S}quamous {C}ell {C}arcinoma with
{I}mputed {S}usceptibility to {E}ndocrine {T}herapy.},
journal = {International journal of molecular sciences},
volume = {25},
number = {2},
issn = {1422-0067},
address = {Basel},
publisher = {Molecular Diversity Preservation International},
reportid = {DKFZ-2024-00224},
pages = {1244},
year = {2024},
note = {#LA:E221#},
abstract = {Head and neck squamous cell carcinoma (HNSCC) is associated
with high morbidity and mortality. New personalized
treatment strategies represent an unmet medical need to
improve the overall survival and the quality of life of
patients, which are often limited by the toxicity of
established multimodal treatment protocols. Several studies
have reported an increased expression of the estrogen
receptor 1 (ESR1) in HNSCC, but its potential role in the
disease outcome of these tumors remains elusive. Using an
integrative analysis of multiomics and clinical data from
The Cancer Genome Atlas (TCGA)-HNSC, we established a
prognostic risk model based on an ESR1-related 25-gene set.
The prognostic value was confirmed in an independent cohort
of HNSCC and other solid tumors from TCGA. Finally, we
performed in silico drug sensitivity modeling to explore
potential vulnerabilities for both risk groups. This
approach predicted a higher sensitivity for HNSCC, with
prominent ESR1 pathway activity under treatment with
specific estrogen receptor modulators. In conclusion, our
data confirm the involvement of ESR1-related pathway
activity in the progression of a defined subset of HNSCC,
provide compelling evidence that these tumors share a
specific vulnerability to endocrine therapy, and pave the
way for preclinical studies and clinical trials to
demonstrate the efficacy of this new therapeutic option.},
keywords = {endocrine therapy (Other) / estrogen receptor alpha (Other)
/ head and neck cancers (Other) / risk model (Other)},
cin = {E221},
ddc = {540},
cid = {I:(DE-He78)E221-20160331},
pnm = {315 - Bildgebung und Radioonkologie (POF4-315)},
pid = {G:(DE-HGF)POF4-315},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:38279245},
pmc = {pmc:PMC10816965},
doi = {10.3390/ijms25021244},
url = {https://inrepo02.dkfz.de/record/287409},
}