TY - JOUR
AU - Ramesh, Palaniappan
AU - Al Kadi, Amal R
AU - Borse, Gaurav M
AU - Webendörfer, Maximilian
AU - Zaun, Gregor
AU - Metzenmacher, Martin
AU - Doerr, Fabian
AU - Bölükbas, Servet
AU - Hegedüs, Balazs
AU - Lueong, Smiths S
AU - Magne, Joelle
AU - Liu, Beiyun
AU - Nunez, Greisly
AU - Schuler, Martin
AU - Green, Douglas R
AU - Kalkavan, Halime
TI - BCL-B Promotes Lung Cancer Invasiveness by Direct Inhibition of BOK.
JO - Cells
VL - 14
IS - 4
SN - 2073-4409
CY - Basel
PB - MDPI
M1 - DKFZ-2025-00446
SP - 246
PY - 2025
AB - Expression of BCL-B, an anti-apoptotic BCL-2 family member, is correlated with worse survival in lung adenocarcinomas. Here, we show that BCL-B can mitigate cell death initiation through interaction with the effector protein BOK. We found that this interaction can promote sublethal mitochondrial outer membrane permeabilization (MOMP) and consequently generate apoptosis-flatliners, which represent a source of drug-tolerant persister cells (DTPs). The engagement of endothelial-mesenchymal-transition (EMT) further promotes cancer cell invasiveness in such DTPs. Our results reveal that BCL-B fosters cancer cell aggressiveness by counteracting complete MOMP.
KW - Humans
KW - Lung Neoplasms: pathology
KW - Lung Neoplasms: metabolism
KW - Lung Neoplasms: genetics
KW - Neoplasm Invasiveness
KW - Proto-Oncogene Proteins c-bcl-2: metabolism
KW - Apoptosis
KW - Cell Line, Tumor
KW - Epithelial-Mesenchymal Transition: genetics
KW - Mitochondrial Membranes: metabolism
KW - BCL-2 family (Other)
KW - BCL-B (Other)
KW - BOK (Other)
KW - DTP (Other)
KW - EMT (Other)
KW - cancer (Other)
KW - drug-resistance (Other)
KW - invasiveness (Other)
KW - mitochondrial permeabilization (Other)
KW - persister phenotype (Other)
KW - Proto-Oncogene Proteins c-bcl-2 (NLM Chemicals)
LB - PUB:(DE-HGF)16
C6 - pmid:39996719
C2 - pmc:PMC11853756
DO - DOI:10.3390/cells14040246
UR - https://inrepo02.dkfz.de/record/299486
ER -