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@ARTICLE{Kool:127641,
author = {M. Kool$^*$ and D. Jones$^*$ and N. Jäger$^*$ and P. A.
Northcott$^*$ and T. J. Pugh and V. Hovestadt$^*$ and R. M.
Piro$^*$ and L. A. Esparza and S. L. Markant and M. Remke
and T. Milde and F. Bourdeaut and M. Ryzhova and D.
Sturm$^*$ and E. Pfaff$^*$ and S. Stark$^*$ and S.
Hutter$^*$ and H. Seker-Cin$^*$ and P. Johann$^*$ and S.
Bender$^*$ and C. Schmidt$^*$ and T. Rausch and D. Shih and
J. Reimand and L. Sieber$^*$ and A. Wittmann$^*$ and L.
Linke$^*$ and H. Witt$^*$ and U. Weber$^*$ and M.
Zapatka$^*$ and R. König$^*$ and R. Beroukhim and G.
Bergthold and P. van Sluis and R. Volckmann and J. Koster
and R. Versteeg and S. Schmidt$^*$ and S. Wolf$^*$ and C.
Lawerenz$^*$ and C. C. Bartholomae$^*$ and C. von Kalle$^*$
and A. Unterberg and C. Herold-Mende and S. Hofer and A. E.
Kulozik and A. von Deimling$^*$ and W. Scheurlen and J.
Felsberg and G. Reifenberger and M. Hasselblatt and J. R.
Crawford and G. A. Grant and N. Jabado and A. Perry and C.
Cowdrey and S. Croul and G. Zadeh and J. O. Korbel and F.
Doz and O. Delattre and G. D. Bader and M. G. McCabe and V.
P. Collins and M. W. Kieran and Y.-J. Cho and S. L. Pomeroy
and O. Witt$^*$ and B. Brors$^*$ and M. D. Taylor and U.
Schüller and A. Korshunov$^*$ and R. Eils$^*$ and R. J.
Wechsler-Reya and P. Lichter$^*$ and S. Pfister$^*$},
collaboration = {I. P. T. Project},
title = {{G}enome sequencing of {SHH} medulloblastoma predicts
genotype-related response to smoothened inhibition.},
journal = {Cancer cell},
volume = {25},
number = {3},
issn = {1535-6108},
address = {Cambridge, Mass.},
publisher = {Cell Press},
reportid = {DKFZ-2017-03664},
pages = {393 - 405},
year = {2014},
abstract = {Smoothened (SMO) inhibitors recently entered clinical
trials for sonic-hedgehog-driven medulloblastoma (SHH-MB).
Clinical response is highly variable. To understand the
mechanism(s) of primary resistance and identify pathways
cooperating with aberrant SHH signaling, we sequenced and
profiled a large cohort of SHH-MBs (n = 133). SHH pathway
mutations involved PTCH1 (across all age groups), SUFU
(infants, including germline), and SMO (adults). Children >3
years old harbored an excess of downstream MYCN and GLI2
amplifications and frequent TP53 mutations, often in the
germline, all of which were rare in infants and adults.
Functional assays in different SHH-MB xenograft models
demonstrated that SHH-MBs harboring a PTCH1 mutation were
responsive to SMO inhibition, whereas tumors harboring an
SUFU mutation or MYCN amplification were primarily
resistant.},
keywords = {Biphenyl Compounds (NLM Chemicals) / GLI2 protein, human
(NLM Chemicals) / Hedgehog Proteins (NLM Chemicals) /
Kruppel-Like Transcription Factors (NLM Chemicals) / LDE225
(NLM Chemicals) / MYCN protein, human (NLM Chemicals) /
N-Myc Proto-Oncogene Protein (NLM Chemicals) / Nuclear
Proteins (NLM Chemicals) / Oncogene Proteins (NLM Chemicals)
/ PTCH protein, human (NLM Chemicals) / Patched Receptors
(NLM Chemicals) / Patched-1 Receptor (NLM Chemicals) / Ptch1
protein, mouse (NLM Chemicals) / Pyridines (NLM Chemicals) /
Receptors, Cell Surface (NLM Chemicals) / Receptors,
G-Protein-Coupled (NLM Chemicals) / Repressor Proteins (NLM
Chemicals) / SHH protein, human (NLM Chemicals) / SMO
protein, human (NLM Chemicals) / SUFU protein, human (NLM
Chemicals) / Smoothened Receptor (NLM Chemicals) / TP53
protein, human (NLM Chemicals) / Tumor Suppressor Protein
p53 (NLM Chemicals) / Phosphatidylinositol 3-Kinases (NLM
Chemicals) / Proto-Oncogene Proteins c-akt (NLM Chemicals) /
TERT protein, human (NLM Chemicals) / Telomerase (NLM
Chemicals) / DDX3X protein, human (NLM Chemicals) / DEAD-box
RNA Helicases (NLM Chemicals)},
cin = {B062 / B080 / B060 / G100 / G380 / G340 / W190},
ddc = {610},
cid = {I:(DE-He78)B062-20160331 / I:(DE-He78)B080-20160331 /
I:(DE-He78)B060-20160331 / I:(DE-He78)G100-20160331 /
I:(DE-He78)G380-20160331 / I:(DE-He78)G340-20160331 /
I:(DE-He78)W190-20160331},
pnm = {312 - Functional and structural genomics (POF3-312)},
pid = {G:(DE-HGF)POF3-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:24651015},
pmc = {pmc:PMC4493053},
doi = {10.1016/j.ccr.2014.02.004},
url = {https://inrepo02.dkfz.de/record/127641},
}