TY - JOUR
AU - Weigel, Christoph
AU - Veldwijk, Marlon R
AU - Oakes, Christopher C
AU - Seibold, Petra
AU - Slynko, Alla
AU - Liesenfeld, David B
AU - Rabionet, Mariona
AU - Hanke, Sabrina
AU - Wenz, Frederik
AU - Sperk, Elena
AU - Benner, Axel
AU - Rösli, Christoph
AU - Sandhoff, Roger
AU - Assenov, Yassen
AU - Plass, Christoph
AU - Herskind, Carsten
AU - Chang-Claude, Jenny
AU - Schmezer, Peter
AU - Popanda, Odilia
TI - Epigenetic regulation of diacylglycerol kinase alpha promotes radiation-induced fibrosis.
JO - Nature Communications
VL - 7
IS - NN
SN - 2041-1723
CY - London
PB - Nature Publishing Group
M1 - DKFZ-2017-05925
SP - 10893 -
PY - 2016
AB - Radiotherapy is a fundamental part of cancer treatment but its use is limited by the onset of late adverse effects in the normal tissue, especially radiation-induced fibrosis. Since the molecular causes for fibrosis are largely unknown, we analyse if epigenetic regulation might explain inter-individual differences in fibrosis risk. DNA methylation profiling of dermal fibroblasts obtained from breast cancer patients prior to irradiation identifies differences associated with fibrosis. One region is characterized as a differentially methylated enhancer of diacylglycerol kinase alpha (DGKA). Decreased DNA methylation at this enhancer enables recruitment of the profibrotic transcription factor early growth response 1 (EGR1) and facilitates radiation-induced DGKA transcription in cells from patients later developing fibrosis. Conversely, inhibition of DGKA has pronounced effects on diacylglycerol-mediated lipid homeostasis and reduces profibrotic fibroblast activation. Collectively, DGKA is an epigenetically deregulated kinase involved in radiation response and may serve as a marker and therapeutic target for personalized radiotherapy.
KW - EGR1 protein, human (NLM Chemicals)
KW - Early Growth Response Protein 1 (NLM Chemicals)
KW - RNA, Messenger (NLM Chemicals)
KW - Diacylglycerol Kinase (NLM Chemicals)
LB - PUB:(DE-HGF)16
C6 - pmid:26964756
C2 - pmc:PMC4792958
DO - DOI:10.1038/ncomms10893
UR - https://inrepo02.dkfz.de/record/130847
ER -