% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Longuespe:285101,
author = {R. Longuespée$^*$ and J. Kunz and M. Fresnais and K. I.
Foerster and J. Burhenne and M. Thomas and D. Kazdal and A.
Stenzinger and P. Christopoulos and W. E. Haefeli},
title = {{T}herapeutic drug monitoring of osimertinib in non-small
cell lung cancer and short bowel syndrome: {A} case report.},
journal = {British journal of clinical pharmacology},
volume = {90},
number = {1},
issn = {0306-5251},
address = {Oxford},
publisher = {Wiley-Blackwell},
reportid = {DKFZ-2023-02225},
pages = {344-349},
year = {2024},
note = {Case report / 2024 Jan;90(1):344-349 / #EA:B350#},
abstract = {Short bowel syndrome (SBS) following extensive intestinal
resection is often characterized by impaired absorption of
orally administered drugs, including tyrosine kinase
inhibitors (TKI). We report the case of a patient with
EGFR-mutated non-small cell lung carcinoma treated with 80
mg/day of the TKI osimertinib who achieved partial response
of the tumour, but was subsequently subjected to a
double-barrelled jejunostomy due to ileus. Due to the
development of SBS after the bypass surgery, plasma
concentrations of osimertinib were monitored using mass
spectrometry. The therapeutic drug monitoring confirmed a
malabsorption of osimertinib in the patient (108 ng/mL,
which is below the 5th percentile of the expected plasma
concentration) and was useful to guide adjustments of TKI
dosing in order to achieve adequate blood levels (161 ng/mL
after increase of the dose to 120 mg/day) in order to
maintain tumour control.},
keywords = {LC-MS/MS (Other) / MALDI-MS/MS (Other) / non-small cell
lung cancer (Other) / osimertinib (Other) / short bowel
syndrome (Other) / therapeutic drug monitoring (Other)},
cin = {B350},
ddc = {610},
cid = {I:(DE-He78)B350-20160331},
pnm = {312 - Funktionelle und strukturelle Genomforschung
(POF4-312)},
pid = {G:(DE-HGF)POF4-312},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:37815301},
doi = {10.1111/bcp.15924},
url = {https://inrepo02.dkfz.de/record/285101},
}